Protease Inhibitors and Phosphatase Inhibitors
MilliporeSigma™ Calbiochem™ 5-Fluorouracil
Potent antitumor agent.
MilliporeSigma™ Calbiochem™ Omeprazole
A cell-permeable pyridyl methylsulfinyl benzimidazole compound that acts as selective proton pump inhibitor.
MilliporeSigma™ Calbiochem™ LFM-A13
A potent, cell-permeable, reversible, substrate competitive, and specific inhibitor of Bruton's Tyrosine Kinase (BTK; IC50 = 17.2μM for human BTK
MilliporeSigma™ Calbiochem™ Kenpaullone
A potent, cell-permeable, and reversible inhibitor of glycogen synthase kinase-3β (IC50 = 230 nM), Lck (IC50 = 470 nM), and cyclin-dependent kinases (Cdks).
MilliporeSigma™ Calbiochem™ MKLP-2 Inhibitor, Paprotrain
The MKLP-2 Inhibitor, Paprotrain controls the biological activity of MKLP-2. This small molecule/inhibitor is primarily used for Cell Signaling applications.
MilliporeSigma™ Calbiochem™ Survivin Antagonist, S12
The Survivin Antagonist, S12 controls the biological activity of Survivin.
MilliporeSigma™ Calbiochem™ Nociceptin
Endogenous ligand for the opioid-like G-protein coupled receptor, ORL1 (Opioid Receptor-Like 1).
MilliporeSigma™ Calbiochem™ 2-N-Hexadecanoylamino-4-nitrophenylphosphorylcholine
Synthetic chromogenic analog of sphingomyelin.
MilliporeSigma™ Calbiochem™ Isradipine
A voltage gated calcium channel gating inhibitor of the dihydropyridine class.
MilliporeSigma™ Calbiochem™ Psalmotoxin-1
A potent proton-gated sodium channel (ASIC1a) channel blocking neurotoxin (IC50 = 0.9 nM) that can distinguish between the two ASIC1 splice variants, ASIC1a and ASIC1b.
MilliporeSigma™ Calbiochem™ NF-κB Activation Inhibitor
The NF-κB Activation Inhibitor, also referenced under CAS 545380-34-5, controls the biological activity of NF-κB. This small molecule/inhibitor is primarily used for Inflammation/Immunology applications.
Thermo Scientific Chemicals Leupeptin, 90%, synthetic
CAS: 103476-89-7 Molecular Formula: 0·5 H2O4S
MilliporeSigma™ Calbiochem™ Gö 6976
Gö 6976, CAS 136194-77-9, is a cell-permeable, reversible, and ATP-competitive inhibitor of PKC (IC50 = 7.9 nM for rat brain). Exhibits selectively for PKCα (IC50 = 2.3 nM) and βI (IC50 = 6.2 nM).
MilliporeSigma™ Calbiochem™ GPR40 Antagonist, GW1100
The GPR40 Antagonist, GW1100, also referenced under CAS 306974-70-9, controls the biological activity of GPR40. This small molecule/inhibitor is primarily used for Biochemicals applications.